SCHEMBL9518147

SCHEMBL9518147

Cc1nc2ccc(C)c(C)c2c(=O)[nH]1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.64
TYMS P04818 15/20 0.58
BMPR1B O00238 1/20 0.52
RAF1 P04049 1/20 0.52
BRAF P15056 1/20 0.52
BMPR1A P36894 1/20 0.52
ACVR1B P36896 1/20 0.52
TGFBR1 P36897 1/20 0.52
ACVRL1 P37023 1/20 0.52
ACVR1 Q04771 1/20 0.52
TNKS2 Q9H2K2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15840744 0.82 PARP1 (0.66) PARP1TYMSBMPR1BRAF1BRAF
SCHEMBL19992076 0.82 PARP1 (0.66) PARP1TYMSBMPR1BRAF1BRAF
SCHEMBL16306348 0.82 PARP1 (0.61) PARP1TYMSTNKS2
SCHEMBL7826334 0.82 PARP1 (0.60) PARP1TYMSTNKS2
SCHEMBL9259148 0.78 PARP1 (1.00) PARP1TYMSBMPR1BRAF1BRAF
SCHEMBL30838794 0.78 PARP1 (1.00) PARP1TYMSBMPR1BRAF1BRAF
SCHEMBL19992101 0.75 PARP1 (0.66) PARP1TYMSBMPR1BRAF1BRAF
SCHEMBL15840736 0.75 PARP1 (0.66) PARP1TYMSBMPR1BRAF1BRAF
SCHEMBL6653100 0.74 TYMS (1.00) PARP1TYMSBMPR1BRAF1BRAF
SCHEMBL7826662 0.73 TYMS (1.00) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284338-B1 Anti-tumour agents ICI PLC (GB) 1993-12-22 EP disclosed
US-4981856-A QUINAZOLINE IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-01 US disclosed
EP-0284338-A2 Anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-09-28 EP disclosed