SCHEMBL951880

SCHEMBL951880

CC(=O)/C=C/N(C)C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15043324 1.00
SCHEMBL951882 1.00
SCHEMBL18752199 0.80 POLB (0.48)
SCHEMBL7345262 0.78 TDP1 (0.52)
SCHEMBL7345258 0.78 TDP1 (0.52)
SCHEMBL13887197 0.77 TDP1 (0.46)
SCHEMBL25246733 0.75
SCHEMBL263813 0.75
SCHEMBL1430406 0.75
SCHEMBL12864549 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 254 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117384096-A Preparation method of difluoro pyrazole acid 山东国邦药业有限公司 2024-01-12 CN claimed
EP-0873746-A2 Dyestuff for keratinous fibers Henkel Kommanditgesellschaft auf Aktien (DE) 1998-10-28 EP claimed
JP-3038583-A None JP disclosed
US-20260116868-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2026-04-30 US disclosed
EP-4720055-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF Arcus Biosciences, Inc. (US) 2026-04-08 EP disclosed
US-20250320213-A1 Nitrogen-Containing Heterocyclic Compounds PFIZER INC. (US) 2025-10-16 US disclosed
WO-2025215579-A1 NOVEL NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS PFIZER INC. (US) 2025-10-16 WO disclosed
WO-2025076299-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2025-04-10 WO disclosed
CN-114008065-B Glycyrrhetinic acid derivatives for the treatment of hyperkalemia 阿德利克斯股份有限公司 2025-03-11 CN disclosed
US-20250011318-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2025-01-09 US disclosed
WO-2024243502-A1 CBL-B INHIBITORS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2024-11-28 WO disclosed
EP-0608725-B1 Process for preparing aminomethylene compounds BAYER AG (DE) 2000-05-17 EP disclosed
EP-0873746-A2 Dyestuff for keratinous fibers Henkel Kommanditgesellschaft auf Aktien (DE) 1998-10-28 EP disclosed
US-5401869-A Process for the preparation of aminomethylene compounds BAYER AKTIENGESELLSCHAFT (DE) 1995-03-28 US disclosed
EP-0406839-B1 Process for the preparation of 1-(4-tetrahydropyranyl) or 1-(4-tetrahydrothiopyranyl)-prop-1-en-3-ones BASF AG (DE) 1995-02-01 EP disclosed
EP-0608725-A2 Process for preparing aminomethylene compounds BAYER AG (DE) 1994-08-03 EP disclosed
US-5221753-A PREPARATION OF 1-(4-TETRAHYDROPYRANYL)- OR 1-(4-TETRAHYDROTHIOPYRANYL)PROP-1-EN-3-ONES BASF AKTIENGESELLSCHAFT (DE) 1993-06-22 US disclosed
JP-H0338583-A PRODUCTION OF 1-(4-TETRAHYDROPYRANYL)-1-BUTEN-3-ONE NIPPON SODA CO LTD 1991-02-19 JP disclosed
EP-0406839-A2 Process for the preparation of 1-(4-tetrahydropyranyl) or 1-(4-tetrahydrothiopyranyl)-prop-1-en-3-ones BASF Aktiengesellschaft (DE) 1991-01-09 EP disclosed
EP-0322616-A2 Novel 5(and/or 6)substituted 2-(2-imidazolin-2-yl)nicotinic acids, esters and salts, useful as herbicidal agents and nivel intermediates for the preparation of said nicotinic acids, esters and salts AMERICAN CYANAMID COMPANY (US) 1989-07-05 EP disclosed