SCHEMBL9519265

SCHEMBL9519265

O=c1[nH]c(-c2ccc(CCCCCl)cc2)cs1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
BRD4 O60885 10/20 0.53
SMN1; SMN2 Q16637 1/20 0.51
GPR84 Q9NQS5 2/20 0.39
CTSV O60911 2/20 0.36
CTSL P07711 2/20 0.36
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
IDO1 P14902 1/20 0.35
PPARG P37231 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
NCOA2 Q15596 1/20 0.35
NCOA1 Q15788 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
S1PR4 O95977 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR5 Q9H228 1/20 0.34
NEK1 Q96PY6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9519379 0.89 ALDH1A1 (0.62) ALDH1A1BRD4SMN1; SMN2GPR84MEN1
Bromide SCHEMBL9518983 0.88 ALDH1A1 (0.60) ALDH1A1BRD4SMN1; SMN2GPR84MEN1
SCHEMBL16414571 0.83 BRD4 (0.54) ALDH1A1BRD4SMN1; SMN2GPR84CTSV
SCHEMBL3836008 0.73 ALDH1A1 (1.00) ALDH1A1BRD4SMN1; SMN2MEN1POLB
SCHEMBL9553269 0.72 HRH3 (0.43) ALDH1A1SMN1; SMN2MEN1MAPTRAB9A
SCHEMBL9552525 0.72 HRH3 (0.43) ALDH1A1SMN1; SMN2MEN1MAPTRAB9A
SCHEMBL16414517 0.70 BRD4 (0.67) ALDH1A1BRD4SMN1; SMN2CTSVCTSL
SCHEMBL16414580 0.70 BRD4 (0.67) ALDH1A1BRD4SMN1; SMN2MEN1POLB
SCHEMBL9135033 0.70 MAOB (0.44) ALDH1A1SMN1; SMN2MAPT
SCHEMBL16415205 0.70 SMN1; SMN2 (0.92) ALDH1A1BRD4SMN1; SMN2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279598-B1 ARYLPIPERAZINYL-ALKYLENE-PHENYL-HETEROCYCLIC COMPOUNDS PFIZER INC. (US) 1993-09-15 EP disclosed
US-4891375-A Arylpiperazinyl-alkylene-phenyl-heterocyclic compounds PFIZER INC. (US) 1990-01-02 US disclosed
EP-0279598-A2 Arylpiperazinyl-alkylene-phenyl-heterocyclic compounds PFIZER INC. (US) 1988-08-24 EP disclosed