SCHEMBL9520221

SCHEMBL9520221

COc1ccc(/C(C)=C/C=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 3/20 0.53
CES2 O00748 2/20 0.52
CES1 P23141 2/20 0.52
CA1 P00915 4/20 0.52
CA2 P00918 4/20 0.52
PTGS1 P23219 1/20 0.51
PTGS2 P35354 1/20 0.51
TCF4 P15884 1/20 0.49
CTNNB1 P35222 1/20 0.49
MAPT P10636 2/20 0.48
PARP1 P09874 1/20 0.48
PARP10 Q53GL7 1/20 0.48
PARP2 Q9UGN5 1/20 0.48
PARP4 Q9UKK3 1/20 0.48
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4962948 1.00 NQO2 (0.53) NQO2CES2CES1CA1CA2
SCHEMBL3071944 1.00 NQO2 (0.53) NQO2CES2CES1CA1CA2
SCHEMBL19659965 0.85 NQO2 (0.44) NQO2CES2CES1CA1CA2
SCHEMBL8564034 0.82 ALDH1A1 (0.57) NQO2CES2CES1CA1CA2
SCHEMBL24181271 0.80 NQO2 (0.53) NQO2CES2CES1CA1CA2
SCHEMBL6554966 0.80 NQO2 (0.44) NQO2PTGS1ALDH1A1KDM4E
SCHEMBL2472466 0.80 NQO2 (0.61) NQO2PTGS1PTGS2MAPTALDH1A1
SCHEMBL6554972 0.80 NQO2 (0.44) NQO2PTGS1ALDH1A1KDM4E
SCHEMBL8428783 0.79 NQO2 (0.56) NQO2CES2CES1CA1CA2
SCHEMBL8428781 0.79 NQO2 (0.56) NQO2CES2CES1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112321544-B Chiral quaternary carbon cyanide and preparation method thereof 深圳湾实验室坪山生物医药研发转化中心 2023-05-26 CN disclosed
WO-2022127712-A1 METHOD FOR STEREOSPECIFIC SYNTHESIS OF 2-ENAL AND 2-ENONE COMPOUNDS, AND DEUTERATED COMPOUNDS THEREOF 复旦大学 2022-06-23 WO disclosed
CN-106414392-B 6,7,8, 9-tetrahydro-5H-benzo [7] annulene-2-alkylamine compound and application thereof 华东理工大学 2019-05-14 CN disclosed
CN-108117534-A The oxygen-containing cycloaliphatic ring methylamines of benzo 华东理工大学 2018-06-05 CN disclosed
CN-108084125-A Benzheterocycle alkyl amine compound and application thereof 华东理工大学 2018-05-29 CN disclosed
CN-107531613-A Benzo cycloaliphatic ring substituted alkylamine class compound and application thereof 华东理工大学 2018-01-02 CN disclosed
CN-105566262-B Alkyl amine compound of benzofuran 7 and application thereof 华东理工大学 2017-10-27 CN disclosed
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed
US-4788206-A CARDIOVASCULAR DISORDERS, PLATELETS HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed