SCHEMBL9520230

SCHEMBL9520230

C=CCOC(=O)N1C[C@H](OS(C)(=O)=O)C[C@H]1COCC(=O)NC(N)=O

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.33
ANPEP P15144 1/20 0.33
MAPT P10636 1/20 0.30
CACNA1B Q00975 1/20 0.30
APBA1 Q02410 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9519472 0.85 MMP2 (0.30) MMP2ANPEP
SCHEMBL9519285 0.85 MMP2 (0.30) MMP2ANPEP
SCHEMBL9374200 0.83 CYP19A1 (0.32) MMP2ANPEP
SCHEMBL9374194 0.83 CYP19A1 (0.32) MMP2ANPEP
SCHEMBL10518534 0.83
SCHEMBL9794948 0.83
SCHEMBL9519206 0.82 ITGB1 (0.40) MAPT
SCHEMBL9429298 0.82
SCHEMBL9520725 0.81 MAPT (0.34) MAPTCACNA1BAPBA1
SCHEMBL9795047 0.80 CYP19A1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0280771-B1 3-Pyrrolidinylthio-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid derivatives and processes for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-07-28 EP disclosed
US-5061804-A 3-thiopyrrolidine as chemical intermediates FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-10-29 US disclosed
US-4963543-A BACTERICIDES, TREATING INFECTIOUS DISEASES; THIENAMYCINS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-10-16 US disclosed
EP-0280771-A1 3-Pyrrolidinylthio-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid derivatives and processes for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-09-07 EP disclosed