Bicarbonate

Bicarbonate

SCHEMBL9520341

Brc1ccc(CCCCCc2cccnc2)cc1.O=C(O)O

nearest known ligand 0.66

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 9/20 0.66
CHRNA7 P36544 1/20 0.57
HRH1 P35367 2/20 0.55
TDP1 Q9NUW8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
CYP2A6 P11509 1/20 0.50
NAPRT Q6XQN6 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
PTAFR P25105 2/20 0.49
TRPV1 Q8NER1 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL9522433 0.89 TBXAS1 (0.81) TBXAS1CHRNA7HRH1TDP1L3MBTL1
SCHEMBL13098626 0.82 HRH1 (0.72) TBXAS1CHRNA7HRH1TDP1L3MBTL1
SCHEMBL12040598 0.82 HRH1 (0.72) TBXAS1CHRNA7HRH1TDP1L3MBTL1
Bicarbonate SCHEMBL9522368 0.81 TDP1 (0.81) TBXAS1HRH1TDP1L3MBTL1CYP2A6
Bicarbonate SCHEMBL9520058 0.81 TDP1 (0.81) TBXAS1HRH1TDP1L3MBTL1CYP2A6
Bicarbonate SCHEMBL9520418 0.81 TDP1 (0.81) TBXAS1HRH1TDP1L3MBTL1CYP2A6
SCHEMBL8199794 0.80 TDP1 (0.71) TBXAS1CHRNA7HRH1TDP1L3MBTL1
SCHEMBL9520336 0.80 TBXAS1 (0.53) TBXAS1CHRNA7HRH1TDP1L3MBTL1
SCHEMBL8658187 0.80 HRH1 (0.81) TBXAS1CHRNA7HRH1TDP1L3MBTL1
SCHEMBL2845851 0.80 HRH1 (0.81) TBXAS1CHRNA7HRH1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed