SCHEMBL9520378

SCHEMBL9520378

N=C(Nc1ccccc1)N1CCOCC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.65
CYP2C9 P11712 1/20 0.65
MAPT P10636 5/20 0.63
NPSR1 Q6W5P4 2/20 0.63
GAA P10253 5/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
HPGD P15428 1/20 0.58
LMNA P02545 2/20 0.55
ALDH1A1 P00352 5/20 0.54
POLB P06746 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HIF1A Q16665 1/20 0.48
EPAS1 Q99814 1/20 0.48
FAAH O00519 1/20 0.47
MGLL Q99685 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HTT P42858 1/20 0.47
PIK3CA P42336 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL10827455 0.98 CYP2C19 (0.63) CYP2C19CYP2C9MAPTNPSR1GAA
SCHEMBL8391995 0.83 ALDH1A1 (0.55) CYP2C19CYP2C9MAPTNPSR1SMN1; SMN2
SCHEMBL8518308 0.83 ALDH1A1 (0.59) CYP2C19CYP2C9MAPTGAASMN1; SMN2
SCHEMBL11165050 0.83 ALDH1A1 (0.53) CYP2C19CYP2C9MAPTNPSR1GAA
SCHEMBL11473652 0.83 SMN1; SMN2 (0.55) MAPTGAASMN1; SMN2HPGDLMNA
Iodide SCHEMBL10827369 0.81 ALDH1A1 (0.58) CYP2C19CYP2C9MAPTGAASMN1; SMN2
Hydrochloric Acid SCHEMBL11483908 0.81 KMT2A (0.58) CYP2C19CYP2C9MAPTGAASMN1; SMN2
SCHEMBL14448354 0.81 ALDH1A1 (0.60) MAPTNPSR1GAASMN1; SMN2HPGD
SCHEMBL10785302 0.81 MAPT (0.56) CYP2C19CYP2C9MAPTLMNAALDH1A1
Iodide SCHEMBL10827361 0.80 ALDH1A1 (0.61) CYP2C19MAPTGAASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0248586-B1 PROCESS FOR PRODUCING AMIDINE SULFONIC ACID INTERMEDIATES FOR GUANIDINES McNeilab, Inc. (US) 1993-08-25 EP disclosed
US-4851094-A OXIDIZING A THIOUREA WITH HYDROGEN PEROXIDE USING A MOLYBDENUM -CONTAINING CATALYST MCNEILAB, INC. (US) 1989-07-25 US disclosed
US-4781866-A Process for producing amidine sulfonic acid intermediates for guanidines MCNEILAB, INC. (US) 1988-11-01 US disclosed
EP-0248586-A2 Process for producing amidine sulfonic acid intermediates for guanidines McNeilab, Inc. (US) 1987-12-09 EP disclosed
US-4693850-A Methane sulfonic acid derivatives MCNEILAB, INC. (US) 1987-09-15 US disclosed
US-4656291-A OXIDIZING THIOUREA DERIVATIVE WITH HYDROGEN PEROXIDE IN PRESENCE OF MOLYBDENUM CATALYST MCNEILAB, INC. (US) 1987-04-07 US disclosed
US-4656270-A Process for producing guanidines such as linogliride MCNEILAB, INC. (US) 1987-04-07 US disclosed
EP-0195620-A2 Process for producing guanidines such as linogliride and process for intermediates McNeilab, Inc. (US) 1986-09-24 EP disclosed