SCHEMBL9520767

SCHEMBL9520767

COc1ccc(CCCC(N)Cc2ccc(O)c3[nH]c(=O)sc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 18/20 0.47
ADRB1 P08588 12/20 0.45
ADRA1D P25100 5/20 0.45
DRD2 P14416 5/20 0.45
DRD3 P35462 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707082 0.81 ADRB2 (0.52) ADRB2ADRB1ADRA1DDRD2DRD3
SCHEMBL9520760 0.80 ADRB2 (0.66) ADRB2ADRB1ADRA1DDRD2DRD3
Hydrochloric Acid SCHEMBL8881126 0.79 ADRB2 (0.65) ADRB2ADRB1ADRA1DDRD2DRD3
SCHEMBL9522342 0.78 ADRB2 (0.72) ADRB2ADRB1ADRA1DDRD2DRD3
SCHEMBL7839170 0.76 ADRB2 (0.46) ADRB2ADRB1DRD2
SCHEMBL7838618 0.75 ADRB2 (0.38) ADRB2ADRB1DRD2DRD3
SCHEMBL7839902 0.75 ADRB2 (0.55) ADRB2ADRB1ADRA1DDRD2
Trifluoroacetic Acid SCHEMBL7839611 0.74 ADRB2 (0.46) ADRB2ADRB1DRD2
SCHEMBL9520825 0.73 ADRB2 (0.55) ADRB2ADRB1DRD2
SCHEMBL1803587 0.73 ADRB2 (0.51) ADRB2ADRB1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558677-A1 BIOLOGICALLY ACTIVE AMINES Astra Pharmaceuticals Limited (GB) 1993-09-08 EP claimed
WO-1992008708-A1 BIOLOGICALLY ACTIVE AMINES FISONS PLC (GB) 1992-05-29 WO claimed