SCHEMBL9522969

SCHEMBL9522969

COC1C[C@H](OCc2ccccc2)[C@@H](OC(C)=O)[C@@H](COC(C)=O)O1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.51
LMNA P02545 2/20 0.50
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 4/20 0.45
CYP2D6 P10635 2/20 0.45
MAPK1 P28482 1/20 0.45
POLB P06746 1/20 0.45
CA12 O43570 6/20 0.42
CA1 P00915 6/20 0.42
CA2 P00918 6/20 0.42
CA9 Q16790 6/20 0.42
CYP3A4 P08684 2/20 0.40
MAPT P10636 1/20 0.40
CA4 P22748 4/20 0.40
CA6 P23280 4/20 0.40
CA5A P35218 4/20 0.40
CA7 P43166 4/20 0.40
CA13 Q8N1Q1 4/20 0.40
CA14 Q9ULX7 4/20 0.40
CA5B Q9Y2D0 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10429257 1.00 TSHR (0.51) TSHRLMNAKMT2AALDH1A1CYP2D6
SCHEMBL23742936 0.89 TSHR (0.53) TSHRLMNAKMT2AALDH1A1CYP2D6
SCHEMBL12573457 0.83 LMNA (0.47) TSHRLMNAKMT2AALDH1A1CYP2D6
SCHEMBL6256354 0.81 CA12 (0.58) TSHRLMNACYP2D6CA12CA1
SCHEMBL19772733 0.81 CA12 (0.58) TSHRLMNACYP2D6CA12CA1
SCHEMBL9684068 0.81 CA12 (0.58) TSHRLMNACYP2D6CA12CA1
SCHEMBL9684071 0.81 CA12 (0.58) TSHRLMNACYP2D6CA12CA1
SCHEMBL25651657 0.81 CA12 (0.58) TSHRLMNACYP2D6CA12CA1
SCHEMBL9094454 0.81 NT5E (0.46) PTPN1
SCHEMBL9094458 0.81 NT5E (0.46) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0302253-B1 3-DEMETHYL-4-FLUORO-MEVALONIC-ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL PREPARATIONS BASED ON THOSE COMPOUNDS, THEIR USE AND INTERMEDIATES HOECHST AKTIENGESELLSCHAFT (DE) 1993-04-07 EP disclosed
US-4898868-A ANTICHOLESTEROL AGENTS; LACTONE OR FREE ACID FORM HOECHST AKTIENGESELLSCHAFT (DE) 1990-02-06 US disclosed