SCHEMBL9523344

SCHEMBL9523344

Cc1cc(N)ccc1NC(=O)OCc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.70
RAB9A P51151 1/20 0.70
MAPT P10636 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
MGLL Q99685 2/20 0.53
FAAH O00519 1/20 0.53
OPRK1 P41145 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
MAOB P27338 1/20 0.49
PLAU P00749 1/20 0.48
POLB P06746 1/20 0.48
CASP3 P42574 1/20 0.47
BLK P51451 1/20 0.47
BTK Q06187 1/20 0.47
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28859639 0.89 NPC1 (0.70) NPC1RAB9AMAPTMGLLFAAH
SCHEMBL6067806 0.85 NPC1 (0.64) NPC1RAB9AMAPTMGLLFAAH
SCHEMBL9524957 0.85 F10 (0.56) NPC1RAB9AMAPTMGLLSMN1; SMN2
SCHEMBL9524227 0.84 NPC1 (0.56) NPC1RAB9AMAPTMGLLFAAH
SCHEMBL1554137 0.84 NPC1 (0.70) NPC1RAB9AMAPTMGLLFAAH
SCHEMBL14648942 0.84 NPC1 (0.70) NPC1RAB9AMAPTCYP1A2CYP2C9
SCHEMBL4201821 0.84 NPC1 (0.66) NPC1RAB9AMAPTMGLLFAAH
SCHEMBL13193092 0.84 RAB9A (0.55) NPC1RAB9AMAPTMGLLHDAC3
SCHEMBL16088310 0.83 NPC1 (0.61) NPC1RAB9AMAPTCYP1A2CYP2C9
SCHEMBL2069644 0.83 SMN1; SMN2 (0.73) MAPTCYP1A2CYP2C9CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0285000-B1 CHROMOGENE COMPOUNDS, THEIR MANUFACTURE AND USE AS ENZYME SUBSTRATES Roche Diagnostics GmbH (DE) 1993-07-28 EP disclosed
US-5190862-A Peptide modified compound BOEHRINGER MANNHEIM GMBH (DE) 1993-03-02 US disclosed
US-5108890-A Diagnostic agents for determining peptide bond-cleaving enzymes; measuring light absorbed by liberated colored materials BOEHRINGER MANNHEIM GMBH (DE) 1992-04-28 US disclosed
EP-0285000-A2 Chromogene compounds, their manufacture and use as enzyme substrates Roche Diagnostics GmbH (DE) 1988-10-05 EP disclosed