SCHEMBL9523733

SCHEMBL9523733

c1ccc(CN2CCOC(c3ccccc3)C2)cc1

nearest known ligand 0.77

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 17/20 0.77
MOGAT2 Q3SYC2 1/20 0.61
DRD4 P21917 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27405274 1.00 CNR2 (0.77) CNR2MOGAT2DRD4
Hydrochloric Acid SCHEMBL8097089 0.98 CNR2 (0.75) CNR2MOGAT2DRD4
SCHEMBL2294156 0.91 CNR2 (0.66) CNR2MOGAT2DRD4
SCHEMBL2294344 0.91 CNR2 (0.66) CNR2MOGAT2DRD4
SCHEMBL82233 0.90 CNR2 (0.64) CNR2MOGAT2DRD4
SCHEMBL2298286 0.90 CNR2 (0.64) CNR2MOGAT2DRD4
SCHEMBL4599689 0.90 CNR2 (0.64) CNR2MOGAT2DRD4
SCHEMBL323333 0.90 CNR2 (0.64) CNR2MOGAT2DRD4
SCHEMBL1438014 0.90 CNR2 (0.64) CNR2MOGAT2DRD4
SCHEMBL4480485 0.90 CNR2 (0.72) CNR2MOGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507863-A4 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF 1993-07-07 EP claimed
EP-0507863-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1992-10-14 EP claimed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO claimed
CN-1106390-C Polymorphic form of tachykinin receptor antagonist 2-(R)-(1-(R)-(3,5-bis(trifluoromethyl) phenyl) ethoxy)-3-(S)-(4-fluoro) phenyl-4-(3-5(oxo-1H,4H-1,2,4-triazolo methylmorpholine MERCK & CO INC (US) 2003-04-23 CN disclosed