SCHEMBL9524355

SCHEMBL9524355

Cc1ccc(C(=O)N2CCN(C(=O)c3ccc(-n4ccnc4)cc3)CC2)nc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.54
TDP1 Q9NUW8 2/20 0.53
CYP3A4 P08684 1/20 0.50
BAZ2B Q9UIF8 1/20 0.50
MAOB P27338 1/20 0.48
HTT P42858 2/20 0.47
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
KMT2A Q03164 2/20 0.46
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
SLC6A7 Q99884 1/20 0.46
ADH5 P11766 2/20 0.45
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9363641 0.80 HPGD (0.68) LSSCYP3A4BAZ2BHTTHTR2A
Hydrochloric Acid SCHEMBL9368954 0.79 HPGD (0.66) LSSCYP3A4BAZ2BHTTHTR2A
SCHEMBL8536306 0.75 LSS (0.60) LSSCYP3A4BAZ2BMAOBHTT
Hydrochloric Acid SCHEMBL5734554 0.74 LSS (0.59) LSSCYP3A4BAZ2BMAOBHTT
SCHEMBL8536934 0.74 HTR2A (0.60) LSSCYP3A4BAZ2BHTTHTR2A
SCHEMBL8537654 0.73 HTR2A (0.59) LSSCYP3A4BAZ2BHTTHTR2A
SCHEMBL20160906 0.73 TDP1 (0.66) TDP1SMN1; SMN2
Hydrochloric Acid SCHEMBL8537801 0.73 HTR2A (0.59) LSSCYP3A4BAZ2BHTTHTR2A
SCHEMBL10329801 0.73 TDP1 (0.65) TDP1HTTSMN1; SMN2HPGD
SCHEMBL46306 0.73 TDP1 (0.65) TDP1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537201-A1 IMIDAZOLYLBENZOYL SUBSTITUTED HETEROCYCLES SCHERING AKTIENGESELLSCHAFT (DE) 1993-04-21 EP disclosed
US-5189036-A Cardiovascular agents; class III antiarrhythmic agents SCHERING AG (DE) 1993-02-23 US disclosed
WO-1991019709-A1 IMIDAZOLYLBENZOYL SUBSTITUTED HETEROCYCLES SCHERING AKTIENGESELLSCHAFT BERLIN UND BERGKAMEN (DE) 1991-12-26 WO disclosed