SCHEMBL9524757

SCHEMBL9524757

CC(C)(C)OC(=O)NCCOC(=O)C1NCCc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
IDO1 P14902 1/20 0.46
OPRM1 P35372 12/20 0.43
NAMPT P43490 1/20 0.41
OPRK1 P41145 4/20 0.40
DRD2 P14416 1/20 0.39
SLC18A2 Q05940 1/20 0.39
MALT1 Q9UDY8 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
OPRD1 P41143 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526031 0.94 TSHR (0.43) TSHRNPSR1IDO1OPRM1NAMPT
SCHEMBL10401735 0.85 TSHR (0.44) TSHRNPSR1OPRM1OPRK1DRD2
SCHEMBL9526040 0.83 TSHR (0.42) TSHRNPSR1IDO1OPRM1OPRK1
SCHEMBL30829405 0.81 TSHR (0.60) TSHRNPSR1OPRM1OPRK1SLC6A2
SCHEMBL7694988 0.81 TSHR (0.60) TSHRNPSR1OPRM1OPRK1SLC6A2
SCHEMBL30442509 0.81 TSHR (0.60) TSHRNPSR1OPRM1OPRK1SLC6A2
SCHEMBL9525510 0.81 TSHR (0.39) TSHRNPSR1OPRM1OPRK1SLC18A2
SCHEMBL9526410 0.78 TSHR (0.58) TSHRNPSR1OPRM1SLC18A2SLC6A2
SCHEMBL9524766 0.77 TSHR (0.47) TSHRNPSR1IDO1OPRM1OPRK1
SCHEMBL9525257 0.77 TSHR (0.47) TSHRNPSR1OPRM1OPRK1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed