SCHEMBL9525568

SCHEMBL9525568

O=C(NCCCCOC(=O)Nc1cccc2ccccc12)OCCN(C(=O)c1cncc(Br)c1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
HPGD P15428 1/20 0.40
LMNA P02545 1/20 0.39
POLB P06746 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TRPV1 Q8NER1 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
KDM4E B2RXH2 2/20 0.36
KDM6B O15054 2/20 0.36
KDM4C Q9H3R0 2/20 0.36
BLM P54132 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KDM4A O75164 1/20 0.36
EGLN2 Q96KS0 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525208 0.99 ALDH1A1 (0.40) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9524400 0.98 ALDH1A1 (0.41) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9528356 0.93 ALDH1A1 (0.41) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9524184 0.93 ALDH1A1 (0.47) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9525424 0.92 ALDH1A1 (0.43) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9525336 0.91 ALDH1A1 (0.40) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9525296 0.88 ALDH1A1 (0.43) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9526036 0.88 ALDH1A1 (0.43) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9524016 0.87 ALDH1A1 (0.41) ALDH1A1HPGDLMNAPOLBNPC1
SCHEMBL9525236 0.87 ALDH1A1 (0.40) ALDH1A1HPGDLMNAPOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed