SCHEMBL9525663

SCHEMBL9525663

CC(c1ccc2[nH]nnc2c1)n1ccnc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 9/20 0.52
CYP26A1 O43174 2/20 0.48
CYP11B1 P15538 4/20 0.44
CYP11B2 P19099 4/20 0.44
CYP19A1 P11511 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9078558 0.82 CYP19A1 (0.60) CYP17A1CYP26A1CYP11B1CYP11B2CYP19A1
Hydrochloric Acid SCHEMBL9663513 0.77 CYP17A1 (0.51) CYP17A1CYP26A1CYP11B1CYP11B2CYP19A1
SCHEMBL27274843 0.77 CYP17A1 (0.51) CYP17A1CYP26A1CYP11B1CYP11B2CYP19A1
SCHEMBL19054891 0.77 CYP17A1 (0.54) CYP17A1CYP26A1CYP11B1CYP11B2CYP19A1
Hydrochloric Acid SCHEMBL9664030 0.76 CYP17A1 (0.53) CYP17A1CYP26A1CYP11B1CYP11B2CYP19A1
SCHEMBL242516 0.75 EIF4A3 (0.39)
SCHEMBL9662820 0.73 CYP17A1 (0.52) CYP17A1CYP26A1CYP11B1CYP11B2CYP19A1
SCHEMBL9662043 0.73 CYP17A1 (0.50) CYP17A1CYP26A1CYP11B1CYP11B2
SCHEMBL11659128 0.72
SCHEMBL21104304 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293978-B1 (1H-AZOL-1-YLMETHYL)SUBSTITUTED BENZOTRIAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-09-15 EP disclosed
US-5039677-A Estrogen inhibitor JANSSEN PHARMACEUTICA N.V. (CA) 1991-08-13 US disclosed
US-4943574-A AROMATASE INHIBITORS, ESTROGEN DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 1990-07-24 US disclosed