SCHEMBL9525904

SCHEMBL9525904

O=Cc1c2ccccc2cc2ccsc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.47
ERN1 O75460 3/20 0.43
MAPT P10636 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2D6 P10635 1/20 0.37
ALOX5 P09917 1/20 0.36
AMY1A P0DUB6 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 2/20 0.35
PADI4 Q9UM07 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779150 0.84 CYP2A6 (0.42) CYP2A6ERN1MAPTCYP1A2CYP2C19
SCHEMBL342278 0.79 ERN1 (0.57) CYP2A6ERN1MAPTCYP1A2CYP2C19
SCHEMBL29388184 0.79 ERN1 (0.57) CYP2A6ERN1MAPTCYP1A2CYP2C19
SCHEMBL9529453 0.76 TUBB4A (0.45) CYP2A6ERN1MAPTCYP1A2CYP2C19
SCHEMBL9526464 0.74 CYP2A6 (0.53) CYP2A6ERN1MAOAMAOBKMT2A
Methyl Alcohol SCHEMBL27670101 0.74 ERN1 (0.57) CYP2A6ERN1MAPTCYP1A2CYP2C19
SCHEMBL10348702 0.73 ERN1 (0.55) CYP2A6ERN1MAPTCYP1A2CYP2C19
SCHEMBL5691810 0.73 PTPN22 (0.41) CYP2A6CYP1A2CYP2C19CYP2D6ALOX5
SCHEMBL4893713 0.72 ERN1 (0.50) CYP2A6ERN1MAPTCYP1A2CYP2C19
SCHEMBL9538077 0.71 CYP2A6 (0.47) CYP2A6ERN1MAPTCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183439-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-02-03 EP disclosed
US-5075455-A Microbiocides, antitumor agents BURROUGHS WELLCOME CO. (US) 1991-12-24 US disclosed
US-5049581-A Dibenzofurans having anti-tumor activity BURROUGHS WELLCOME CO. (US) 1991-09-17 US disclosed
US-5017600-A Antitumor BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5008286-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-04-16 US disclosed
US-4970227-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1990-11-13 US disclosed
US-4866070-A ANTITUMOR AGENT BURROUGHS WELLCOME CO. (US) 1989-09-12 US disclosed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP disclosed