Isoxazole

Isoxazole

SCHEMBL9525946

NC(=O)c1ccsn1.c1cnoc1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
AURKA O14965 1/20 0.32
JAK2 O60674 1/20 0.32
NTRK1 P04629 1/20 0.32
RET P07949 1/20 0.32
PIM1 P11309 1/20 0.32
FGFR1 P11362 1/20 0.32
PRKACA P17612 1/20 0.32
LTK P29376 1/20 0.32
KDR P35968 1/20 0.32
MAP2K2 P36507 1/20 0.32
FLT3 P36888 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
CSNK1A1 P48729 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28835892 0.81 LMNA (0.47) PARP1NPC1LMNARAB9APIM1
SCHEMBL626433 0.81
Hydrochloric Acid SCHEMBL6382691 0.79
Isoxazole SCHEMBL11568599 0.73
Benzamide SCHEMBL3346807 0.71 PARP1 (0.59) PARP1NPC1LMNARAB9AMAPK8
Isoxazole SCHEMBL442195 0.71
Isoxazole SCHEMBL9446168 0.70 PARP1 (0.42) PARP1AURKARETPIM1FGFR1
Isoxazole SCHEMBL22467457 0.69
Isoxazole SCHEMBL8414240 0.67
Isoxazole SCHEMBL9196311 0.66 PARP1 (0.56) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337263-B1 ISOXAZOL(ISOTHIAZOLS)-5-CARBOXAMIDES BASF Aktiengesellschaft (DE) 1993-03-17 EP claimed
EP-0337263-A2 Isoxazol(isothiazols)-5-carboxamides BASF Aktiengesellschaft (DE) 1989-10-18 EP claimed