SCHEMBL9526273

SCHEMBL9526273

COc1ccc2cccc(CCNC(=O)CCl)c2c1

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 17/20 0.82
MTNR1B P49286 8/20 0.81
HTR2C P28335 1/20 0.77
HTR2B P41595 1/20 0.77
NQO2 P16083 2/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29351431 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
SCHEMBL5361538 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
SCHEMBL9490858 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
SCHEMBL9424883 0.89 MTNR1A (0.80) MTNR1AMTNR1BHTR2CHTR2BNQO2
SCHEMBL9492236 0.89 MTNR1A (0.80) MTNR1AMTNR1BHTR2CHTR2BNQO2
SCHEMBL5929467 0.89 MTNR1A (0.87) MTNR1AMTNR1BHTR2CHTR2BNQO2
SCHEMBL12487213 0.89 MTNR1A (0.80) MTNR1AMTNR1BHTR2CHTR2BNQO2
Hydrochloric Acid SCHEMBL9491830 0.88 MTNR1A (0.78) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL114476 0.87 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL1158495 0.87 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0447285-B1 NAPHTHALENE DERIVATIVES, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ADIR ET COMPAGNIE (FR) 1993-05-12 EP claimed
EP-0447285-A1 Naphthalene derivatives, procedure for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-09-18 EP claimed