SCHEMBL9526509

SCHEMBL9526509

CCCCNC(=O)COc1ccc(C2=NNC(=O)CC2)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.51
NPY1R P25929 1/20 0.51
NPY2R P49146 1/20 0.51
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PDE4B Q07343 2/20 0.47
PDE3B Q13370 2/20 0.47
PDE3A Q14432 2/20 0.47
PDE4A P27815 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
HPGD P15428 2/20 0.45
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
THRB P10828 1/20 0.41
HTT P42858 1/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10475455 0.89 HPGD (0.49) LMNANPY1RNPY2RNPC1RAB9A
SCHEMBL7337123 0.88 PDE3B (0.46) LMNANPY1RNPY2RNPC1RAB9A
SCHEMBL10723099 0.88 HRH3 (0.48) LMNANPC1RAB9ASMN1; SMN2PDE4B
SCHEMBL10867608 0.85 PDE4B (0.48) LMNANPY1RNPY2RNPC1RAB9A
SCHEMBL10474558 0.84 BCHE (0.50) LMNANPC1RAB9ASMN1; SMN2PDE4B
SCHEMBL10475462 0.84 MAPK1 (0.51) LMNAHPGDALDH1A1MAPK1
SCHEMBL10431523 0.84 HRH3 (0.51) LMNASMN1; SMN2PDE4BPDE3BPDE3A
SCHEMBL4884827 0.84 LMNA (0.46) LMNANPC1RAB9ASMN1; SMN2PDE4B
SCHEMBL7326426 0.83 PDE3B (0.47) LMNANPY1RNPY2RNPC1RAB9A
SCHEMBL7336275 0.83 PDE3B (0.47) LMNANPY1RNPY2RNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0330242-B1 PYRIDAZINONE DERIVATIVES, THEIR PREPARATION AND USE Sankyo Company Limited (JP) 1993-09-22 EP disclosed
US-4914093-A CARDIOVASCULAR DISORDERS SANKYO COMPANY LIMITED (JP) 1990-04-03 US disclosed
EP-0330242-A1 Pyridazinone derivatives, their preparation and use Sankyo Company Limited (JP) 1989-08-30 EP disclosed
EP-0178189-A2 Pyridazinone derivatives, their preparation and use SANKYO COMPANY LIMITED (JP) 1986-04-16 EP disclosed