SCHEMBL9526888

SCHEMBL9526888

COc1c(C)cnc(CSc2nc3cc(OC(F)(F)CF)ccc3[nH]2)c1C

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 3/20 0.66
CYP2C9 P11712 8/20 0.42
CYP2C19 P33261 7/20 0.42
CYP1A2 P05177 6/20 0.42
CYP3A4 P08684 6/20 0.42
CYP2D6 P10635 6/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
ATP1A1 P05023 3/20 0.42
ATP1B1 P05026 3/20 0.42
ATP1A3 P13637 3/20 0.42
ATP1B2 P14415 3/20 0.42
ATP4A P20648 3/20 0.42
ATP1A2 P50993 3/20 0.42
ATP4B P51164 3/20 0.42
ATP1B3 P54709 3/20 0.42
FXYD2 P54710 3/20 0.42
ATP1A4 Q13733 3/20 0.42
KMT2A Q03164 5/20 0.41
WDR5 P61964 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527112 0.92 BRS3 (0.69) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL9526883 0.89 BRS3 (0.66) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL29455226 0.88 BRS3 (0.84) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL662986 0.88 BRS3 (0.84) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL9527448 0.87 BRS3 (0.68) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL31529606 0.86 BRS3 (0.82) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL7929368 0.86 BRS3 (0.82) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
Ufiprazole SCHEMBL7950477 0.86 BRS3 (0.82) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL9527121 0.86 BRS3 (0.69) BRS3CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6879158 0.85 BRS3 (0.59) BRS3CYP2C9CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0134400-B1 FLUOROALKOXYSUBSTITUTED PYRIDYLMETHYLTHIO-(OR SULFINYL-)BENZIMIDAZOLES HAVING A SECRETOLYTIC ACTIVITY Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1993-03-24 EP disclosed