SCHEMBL9528623

SCHEMBL9528623

Cc1ccccc1C(O)c1ccncc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.67
CYP3A4 P08684 2/20 0.43
CYP17A1 P05093 1/20 0.43
CYP19A1 P11511 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
ESR1 P03372 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CHEK2 O96017 1/20 0.40
CYP2C9 P11712 2/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL227491 0.84 GAA (0.65) GAACYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL3858791 0.84 GAA (0.65) GAACYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL28973546 0.84 GAA (0.65) GAACYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL8017822 0.80 GAA (1.00) GAACYP3A4CYP17A1SLC6A2SLC6A4
SCHEMBL8805155 0.80 GAA (0.56) GAACYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL598722 0.79 GAA (0.57) GAACYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL23003623 0.78 CYP3A4 (0.48) GAACYP3A4CYP17A1CYP19A1CYP11B1
SCHEMBL8496291 0.78 GAA (0.54) GAACYP3A4CYP17A1CYP19A1CYP11B1
SCHEMBL23882948 0.78 ACHE (0.49) GAACYP3A4CYP17A1CYP19A1CYP11B1
SCHEMBL23882694 0.78 ACHE (0.49) GAACYP3A4CYP17A1CYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231996-B1 NOVEL AMINO ACID DERIVATIVES NOVO NORDISK A/S (DK) 1993-10-06 EP disclosed
US-4931450-A Amino acid derivatives NOVO INDUSTRI A/S (DK) 1990-06-05 US disclosed
EP-0231996-A2 Novel amino acid derivatives NOVO NORDISK A/S (DK) 1987-08-12 EP disclosed