SCHEMBL9529107

SCHEMBL9529107

CC(CO)(CO)NCc1ccc2sc3ccccc3c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN7 P35236 1/20 0.45
DUSP3 P51452 1/20 0.45
PTPN12 Q05209 1/20 0.45
PTPN22 Q9Y2R2 1/20 0.45
GPR3 P46089 1/20 0.39
SLC2A1 P11166 1/20 0.38
CYP1A2 P05177 2/20 0.38
DHODH Q02127 1/20 0.37
MAPT P10636 3/20 0.36
CYP2D6 P10635 3/20 0.36
CYP2C9 P11712 1/20 0.36
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
PTGIR P43119 1/20 0.35
ALDH1A1 P00352 4/20 0.35
MMP12 P39900 2/20 0.35
MMP13 P45452 2/20 0.35
RAB9A P51151 3/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9526374 0.99 PTPN7 (0.44) PTPN7DUSP3PTPN12PTPN22GPR3
SCHEMBL9535916 0.87 PTPN7 (0.40) PTPN7DUSP3PTPN12PTPN22GPR3
SCHEMBL9779319 0.85 SLC2A1 (0.41) PTPN7DUSP3PTPN12PTPN22SLC2A1
SCHEMBL9536796 0.83 SLC2A1 (0.47) PTPN7DUSP3PTPN12PTPN22SLC2A1
SCHEMBL10682965 0.82 SLC2A1 (0.40) SLC2A1CYP1A2CYP2D6PDCD1CD274
Hydrochloric Acid SCHEMBL10986411 0.81 HTT (0.41) SLC2A1CYP1A2CYP2D6PDCD1CD274
Hydrochloric Acid SCHEMBL10679660 0.81 HTT (0.41) SLC2A1CYP1A2CYP2D6PDCD1CD274
SCHEMBL9779052 0.80 SLC2A1 (0.49) PTPN7DUSP3PTPN12PTPN22SLC2A1
SCHEMBL9754468 0.79 SLC2A1 (0.37) SLC2A1MAPTPDCD1CD274ALDH1A1
SCHEMBL9536888 0.78 SLC2A1 (0.52) PTPN7DUSP3PTPN12PTPN22GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017600-A Antitumor BURROUGHS WELLCOME CO. (US) 1991-05-21 US claimed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP claimed
EP-0183439-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-02-03 EP disclosed
US-5075455-A Microbiocides, antitumor agents BURROUGHS WELLCOME CO. (US) 1991-12-24 US disclosed
US-5049581-A Dibenzofurans having anti-tumor activity BURROUGHS WELLCOME CO. (US) 1991-09-17 US disclosed
US-5017600-A Antitumor BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5008286-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-04-16 US disclosed
US-4970227-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1990-11-13 US disclosed
US-4965285-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-10-23 US disclosed
US-4866070-A ANTITUMOR AGENT BURROUGHS WELLCOME CO. (US) 1989-09-12 US disclosed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP disclosed