SCHEMBL9754468

SCHEMBL9754468

Cn1c2ccc(CNC(C)(CO)CO)cc2c2sc3ccccc3c21

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.37
TP53 P04637 5/20 0.34
MAPT P10636 6/20 0.34
RXFP1 Q9HBX9 3/20 0.34
ALDH1A1 P00352 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ESR1 P03372 3/20 0.32
ESR2 Q92731 3/20 0.32
TRPV1 Q8NER1 1/20 0.32
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9754640 0.99 SLC2A1 (0.36) SLC2A1TP53MAPTRXFP1ALDH1A1
SCHEMBL9529107 0.79 PTPN7 (0.45) SLC2A1MAPTALDH1A1PDCD1CD274
Hydrochloric Acid SCHEMBL9526374 0.78 PTPN7 (0.44) SLC2A1MAPTALDH1A1PDCD1CD274
SCHEMBL9539120 0.74 SLC2A1 (0.39) SLC2A1MAPTALDH1A1NPSR1TRPV1
SCHEMBL9754616 0.74 SLC2A1 (0.39) SLC2A1MAPTRXFP1ALDH1A1CD274
Hydrochloric Acid SCHEMBL9779007 0.73 SLC2A1 (0.38) SLC2A1MAPTALDH1A1NPSR1TRPV1
Hydrochloric Acid SCHEMBL9754584 0.73 SLC2A1 (0.38) SLC2A1MAPTRXFP1ALDH1A1CD274
SCHEMBL10682965 0.73 SLC2A1 (0.40) SLC2A1ALDH1A1PDCD1CD274
SCHEMBL9754534 0.72 ALKBH5 (0.35) SLC2A1MAPTRXFP1ALDH1A1NPSR1
SCHEMBL9536888 0.72 SLC2A1 (0.52) SLC2A1TP53MAPTALDH1A1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0447703-A1 Hetero polycyclic biocidal compounds, their synthesis and intermediates therefor,formulations containing them and their use in medicine THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-25 EP claimed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US claimed
WO-1991014688-A1 HETERO POLYCYCLIC BIOCIDAL COMPOUNDS AND THEIR USE IN MEDECINE THE WELLCOME FOUNDATION LIMITED (GB) 1991-10-03 WO disclosed
EP-0447703-A1 Hetero polycyclic biocidal compounds, their synthesis and intermediates therefor,formulations containing them and their use in medicine THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-25 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed