SCHEMBL9529269

SCHEMBL9529269

COC(=O)c1sc(Cl)cc1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
HSD17B10 Q99714 2/20 0.45
COMT P21964 1/20 0.44
KDM4E B2RXH2 3/20 0.44
NPC1 O15118 1/20 0.44
CASP3 P42574 1/20 0.44
RAB9A P51151 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
LMNA P02545 3/20 0.44
XDH P47989 2/20 0.44
GAA P10253 2/20 0.44
POLB P06746 1/20 0.44
NFKB1 P19838 1/20 0.44
GFER P55789 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28175472 0.82 MAPT (0.44) TSHRMAPTKMT2AHSD17B10KDM4E
SCHEMBL26281532 0.82 KMT2A (0.44) TSHRMAPTKMT2AHSD17B10KDM4E
SCHEMBL14419258 0.81 GAA (0.44) TSHRMAPTKMT2AHSD17B10KDM4E
SCHEMBL20893814 0.81 MAPT (0.42) TSHRMAPTKMT2AHSD17B10COMT
SCHEMBL10566679 0.81 KDM4E (0.60) TSHRMAPTKMT2AHSD17B10KDM4E
SCHEMBL7670938 0.80 TSHR (0.45) TSHRMAPTKMT2AHSD17B10COMT
SCHEMBL577650 0.80 MAPT (0.45) TSHRMAPTKMT2AHSD17B10KDM4E
Hydrochloric Acid SCHEMBL31120455 0.79 KDM4E (0.59) TSHRMAPTKMT2AHSD17B10KDM4E
SCHEMBL28175473 0.79 DAO (0.53) TSHRMAPTKMT2AHSD17B10KDM4E
SCHEMBL11622247 0.79 GSK3B (0.60) MAPTKMT2AHSD17B10KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4665733-A1 AMINO-SUBSTITUTED PYRROLOTRIAZINE DERIVATIVES AS INHIBITORS OF SGK1 Bristol-Myers Squibb Company (US) 2025-12-24 EP disclosed
WO-2024173323-A1 AMINO-SUBSTITUTED PYRROLOTRIAZINE DERIVATIVES AS INHIBITORS OF SGK1 BRISTOL-MYERS SQUIBB COMPANY (US) 2024-08-22 WO disclosed
US-20230348441-A1 BICYCLIC COMPOUND THAT ACTS AS CRBN PROTEIN REGULATOR MEDSHINE DISCOVERY INC. (CN) 2023-11-02 US disclosed
WO-2021047674-A1 BICYCLIC COMPOUND THAT ACTS AS CRBN PROTEIN REGULATOR 南京明德新药研发有限公司 2021-03-18 WO disclosed
CN-1025027-C Organic compounds and their use as pharmaceuticals LILLY SA (ES) 1994-06-15 CN disclosed
EP-0297697-B1 Thiophene-2-carboxamide derivatives and their pharmaceutical use LILLY SA (ES) 1993-12-29 EP disclosed
US-4904686-A 3-ALKOXYTHIOPHENE-2-CARBOXAMIDES; CENTRAL NERVOUS SYSTEM DISORDERS LILLY INDUSTRIES LIMITED (GB) 1990-02-27 US disclosed
CN-1030916-A Organic compound and as the application of medicine LILLY SA (ES) 1989-02-08 CN disclosed
EP-0297697-A1 Thiophene-2-carboxamide derivatives and their pharmaceutical use LILLY S.A. (ES) 1989-01-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348441-A1 BICYCLIC COMPOUND THAT ACTS AS CRBN PROTEIN REGULATOR CRBN, CRKL, NCOR1 TSHR 931/4885MAPT 2404/4885KMT2A 2954/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.