SCHEMBL9529596

SCHEMBL9529596

O=Cc1cc2c(ccc3ccccc32)s1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.59
ALDH1A1 P00352 3/20 0.43
HSD17B10 Q99714 3/20 0.43
TSHR P16473 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HIF1A Q16665 1/20 0.42
CYP1B1 Q16678 1/20 0.42
ERN1 O75460 1/20 0.41
HPRT1 P00492 3/20 0.40
PRNP P04156 1/20 0.39
PAX8 Q06710 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
GPR3 P46089 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29847503 1.00 CYP2A6 (0.59) CYP2A6ALDH1A1HSD17B10TSHRTDP1
SCHEMBL12683511 0.84 CYP2A6 (0.54) CYP2A6ALDH1A1KDM4EGPR3
SCHEMBL9526357 0.76 CYP2A6 (0.56) CYP2A6ALDH1A1HSD17B10TSHRTDP1
SCHEMBL9536471 0.76 CYP2A6 (0.51) CYP2A6ALDH1A1HSD17B10TSHRTDP1
SCHEMBL56884 0.75 CYP2A6 (1.00) CYP2A6ERN1CA1CA2
SCHEMBL29629031 0.75 CYP2A6 (1.00) CYP2A6ERN1CA1CA2
Hydrochloric Acid SCHEMBL31458505 0.73 CYP2A6 (0.96) CYP2A6ERN1CA1CA2
SCHEMBL1105107 0.73 CYP2A6 (0.46) CYP2A6ALDH1A1KDM4E
SCHEMBL25410254 0.72 ALDH1A1 (0.48) CYP2A6ALDH1A1HSD17B10TSHRTDP1
SCHEMBL17934651 0.72 ALDH1A1 (0.48) CYP2A6ALDH1A1HSD17B10TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183439-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-02-03 EP disclosed
US-5075455-A Microbiocides, antitumor agents BURROUGHS WELLCOME CO. (US) 1991-12-24 US disclosed
US-5049581-A Dibenzofurans having anti-tumor activity BURROUGHS WELLCOME CO. (US) 1991-09-17 US disclosed
US-5017600-A Antitumor BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5008286-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-04-16 US disclosed
US-4970227-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1990-11-13 US disclosed
US-4965285-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-10-23 US disclosed
US-4866070-A ANTITUMOR AGENT BURROUGHS WELLCOME CO. (US) 1989-09-12 US disclosed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP disclosed