SCHEMBL9530628

SCHEMBL9530628

Cc1c(-c2ccccc2C(=O)O)cccc1-n1ccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.47
CD274 Q9NZQ7 1/20 0.45
TBXAS1 P24557 1/20 0.44
MYC P01106 4/20 0.43
ADH5 P11766 3/20 0.43
CYP3A4 P08684 4/20 0.42
CYP1A2 P05177 3/20 0.42
CYP2D6 P10635 3/20 0.42
CYP2C19 P33261 3/20 0.42
MAPK1 P28482 2/20 0.42
CYP2C9 P11712 2/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
PMP22 Q01453 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
DHODH Q02127 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980582 0.88 IDO1 (0.49) IDO1TBXAS1MYCADH5CYP3A4
SCHEMBL726313 0.81 IDO1 (0.59) IDO1MYCADH5CYP3A4CYP1A2
SCHEMBL5690863 0.80 MEN1 (0.50) IDO1CD274ADH5CYP3A4CYP1A2
SCHEMBL27636993 0.78 CYP3A4 (0.62) IDO1TBXAS1ADH5CYP3A4MEN1
SCHEMBL5319528 0.78 IDO1 (0.47) IDO1TBXAS1CYP3A4CYP1A2CYP2D6
SCHEMBL9640288 0.77 IDO1 (0.50) IDO1TBXAS1ADH5CYP3A4CYP1A2
SCHEMBL9530614 0.77 IDO1 (0.48) IDO1ADH5CYP3A4CYP1A2CYP2D6
SCHEMBL7780279 0.76 IDO1 (0.49) IDO1TBXAS1ADH5CYP3A4CYP1A2
SCHEMBL16719674 0.76 CYP3A4 (0.45) IDO1TBXAS1ADH5CYP3A4CYP1A2
SCHEMBL4020894 0.75 CYP3A4 (0.56) IDO1CD274CYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0555331-A1 N-SUBSTITUTED IMIDAZOL-2-ONE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS. SEARLE & CO (US) 1993-08-18 EP disclosed