SCHEMBL9532663

SCHEMBL9532663

COC(=O)C1=CC[CH]C=C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA12 O43570 3/20 0.38
CA7 P43166 3/20 0.38
CA9 Q16790 3/20 0.38
CA14 Q9ULX7 3/20 0.38
CHRM3 P20309 2/20 0.35
TSHR P16473 2/20 0.34
LMNA P02545 3/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
THRB P10828 1/20 0.34
CHRM1 P11229 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
BLM P54132 1/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
CYP3A4 P08684 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12978511 0.82 CHRM3 (0.34) CA1CA2CA12CA7CA9
SCHEMBL16810704 0.81
SCHEMBL5114658 0.79 CA12 (0.43) CA1CA2CA12CA7CA9
SCHEMBL27990184 0.78
SCHEMBL16195919 0.78 HDAC2 (0.32) TSHR
SCHEMBL1328632 0.76
SCHEMBL4056562 0.74
SCHEMBL27209677 0.73 TSHR (0.39) CA1CA2CA12CA7CA9
SCHEMBL896075 0.71 CHRM3 (0.39) CA1CA2CA12CA7CA9
SCHEMBL6414618 0.70 TSHR (0.37) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0539372-A1 THERAPEUTIC AGENTS The Boots Company PLC (GB) 1993-05-05 EP disclosed
EP-0006735-A1 Secondary amines, their preparation, pharmaceutical compositions containing them and their use BEECHAM GROUP PLC (GB) 1980-01-09 EP disclosed