SCHEMBL9533130

SCHEMBL9533130

C1=C(COCc2ccccc2)OCCC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37
MAOB P27338 2/20 0.36
MAOA P21397 1/20 0.36
LTA4H P09960 1/20 0.36
IDO1 P14902 1/20 0.34
LMNA P02545 2/20 0.34
DAO P14920 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
AGXT P21549 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9532267 0.90 TSHR (0.54) TSHRCYP3A4ALOX15CYP2C19TAAR1
SCHEMBL29555309 0.80 TSHR (0.60) TSHRTAAR1MAOBMAOAIDO1
SCHEMBL8548090 0.78 MAOB (0.38) MAOBMAOA
SCHEMBL20522561 0.75 MAOB (0.44) TSHRCYP3A4ALOX15CYP2C19MAOB
Oxirane SCHEMBL3317346 0.73 TSHR (0.75) TSHRTAAR1MAOBMAOAIDO1
Cyclohexane SCHEMBL8149682 0.73 TSHR (0.83) TSHRLTA4HIDO1LMNACA1
Fluoride SCHEMBL27427280 0.73 TSHR (0.94) TSHRCYP2C19IDO1LMNACA1
Tetrahydrofuran SCHEMBL28823233 0.72 TSHR (0.65) TSHRALOX15TAAR1LTA4HIDO1
SCHEMBL8701180 0.72 TSHR (0.65) TSHRTAAR1MAOBMAOALTA4H
Dioxane SCHEMBL8701185 0.72 TSHR (0.71) TSHRALOX15TAAR1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0251827-B1 NEW CYCLIC ETHER DERIVATIVES, THEIR PREPARATION AND THEIR USE Sankyo Company Limited (JP) 1993-09-15 EP disclosed
US-4891363-A PLATELET ACTIVATING FACTOR ANTAGONISTS SANKYO COMPANY LIMITED (JP) 1990-01-02 US disclosed
EP-0210804-B1 PHOSPHATE ESTER DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE SANKYO COMPANY LIMITED (JP) 1989-05-10 EP disclosed
US-4794183-A ANTICANCER AGENTS SANKYO COMPANY LIMITED (JP) 1988-12-27 US disclosed
EP-0188384-B1 PHOSPHATE ESTER DERIVATIVES, AND THEIR USE AS ANTI-CANCER AGENTS SANKYO COMPANY LIMITED (JP) 1988-11-17 EP disclosed
EP-0251827-A2 New cyclic ether derivatives, their preparation and their use Sankyo Company Limited (JP) 1988-01-07 EP disclosed
EP-0210804-A1 Phosphate ester derivatives, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1987-02-04 EP disclosed
EP-0188384-A1 Phosphate ester derivatives, and their use as anti-cancer agents SANKYO COMPANY LIMITED (JP) 1986-07-23 EP disclosed