SCHEMBL9533369

SCHEMBL9533369

COc1ccc(C(OC2CCNCC2)c2ccc(OC)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
KDM1A O60341 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
SLC6A2 P23975 2/20 0.41
SLC6A3 Q01959 2/20 0.41
CHRM2 P08172 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
CYP2D6 P10635 1/20 0.41
CHRM1 P11229 1/20 0.41
DRD1 P21728 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRM1 P35372 1/20 0.41
DRD3 P35462 1/20 0.41
KCNH2 Q12809 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
ADRB1 P08588 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9563265 0.94 CHRM2 (0.51) SLC6A2SLC6A3CHRM2HTR1AADRA2A
Fumaric Acid SCHEMBL9353458 0.84 HRH1 (0.48) SLC6A2SLC6A3CHRM2HTR1AADRA2A
SCHEMBL6616012 0.83 SLC6A3 (0.44) SLC6A2SLC6A3CHRM2HTR1AADRA2A
SCHEMBL4190405 0.79 DRD3 (0.55) SLC6A2SLC6A3CYP2D6DRD3MEN1
SCHEMBL6982214 0.79 SLC6A3 (0.55) SLC6A2SLC6A3CHRM2ADRA2ACYP2D6
SCHEMBL1802062 0.79 DRD3 (0.59) SLC6A2SLC6A3CHRM2HTR1AADRA2A
Hydrochloric Acid SCHEMBL11199043 0.78 SLC6A2 (0.56) SLC6A2SLC6A3CHRM2ADRA2ACYP2D6
SCHEMBL9352969 0.78 DRD3 (0.54) SLC6A2SLC6A3CHRM2HTR1AADRA2A
Hydrochloric Acid SCHEMBL2476701 0.77 MAPK1 (0.60) SLC6A2SLC6A3CHRM2HTR1AADRA2A
SCHEMBL942628 0.77 HRH1 (0.66) TDP1KDM1AMAOAMAOBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335586-B1 PIPERIDINE & PIPERAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME UBE INDUSTRIES, LTD. (JP) 1993-06-02 EP disclosed
US-4929618-A ANTIALLERGENS, ANTIHISTAMINES UBE INDUSTRIES, LTD. (JP) 1990-05-29 US disclosed
EP-0335586-A1 Piperidine & piperazine derivatives, process for preparing the same and pharmaceutical compositions containing the same UBE INDUSTRIES, LTD. (JP) 1989-10-04 EP disclosed