SCHEMBL9533488

SCHEMBL9533488

Cn1ncc2c1C[S+]([O-])c1cn[nH]c1-2

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.34
CSNK2A1 P68400 1/20 0.34
PLK3 Q9H4B4 1/20 0.34
ACVR1B P36896 1/20 0.31
TGFBR1 P36897 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535703 0.60 PLK1 (0.61) PLK1CSNK2A1PLK3
SCHEMBL9533873 0.59 PLK1 (0.54) PLK1CSNK2A1PLK3
Hydrochloric Acid SCHEMBL9534437 0.58 PLK1 (0.59) PLK1CSNK2A1PLK3
Hydrochloric Acid SCHEMBL9221777 0.56 PLK1 (0.49) PLK1CSNK2A1PLK3
SCHEMBL22216147 0.56 PLK1 (0.50) PLK1CSNK2A1PLK3
SCHEMBL22980483 0.53 PLK1 (0.79) PLK1CSNK2A1PLK3
SCHEMBL21678222 0.53 PLK1 (0.54) PLK1CSNK2A1PLK3
SCHEMBL21678223 0.53 PLK1 (0.46) PLK1CSNK2A1PLK3
SCHEMBL9221790 0.52 CCNA2 (0.47)
SCHEMBL22349291 0.51 PLK1 (0.62) PLK1CSNK2A1PLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276835-B1 PYRAZOLOTHIOPYRANOPYRAZOLES MERRELL DOW PHARMACEUTICALS INC. (US) 1993-03-17 EP disclosed
EP-0276835-A1 Pyrazolothiopyranopyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734431-A Thiopyranodipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed