SCHEMBL9536847

SCHEMBL9536847

NC(=O)NCCN1CCC(Cc2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.49
SSTR5 P35346 2/20 0.49
NR4A2 P43354 1/20 0.49
POLB P06746 1/20 0.49
HRH1 P35367 5/20 0.48
TACR2 P21452 1/20 0.48
TACR1 P25103 1/20 0.48
RAB9A P51151 1/20 0.47
CYP2D6 P10635 4/20 0.47
CHRM1 P11229 3/20 0.47
MCHR1 Q99705 1/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536956 0.91 KCNH2 (0.49) KCNH2SSTR5NR4A2POLBHRH1
SCHEMBL9536186 0.90 MAPT (0.56) SSTR5POLBTP53
SCHEMBL10550102 0.89 GNRHR (0.51) KCNH2SSTR5NR4A2POLBHRH1
SCHEMBL10547215 0.88 POLB (0.49) KCNH2SSTR5NR4A2POLBHRH1
SCHEMBL10547164 0.87 KCNH2 (0.48) KCNH2SSTR5NR4A2POLBHRH1
SCHEMBL9537582 0.87 TP53 (0.53) POLBTP53
SCHEMBL10552831 0.87 KCNH2 (0.47) KCNH2SSTR5NR4A2HRH1TACR2
Oxalic Acid SCHEMBL10552513 0.87 SSTR5 (0.51) KCNH2SSTR5NR4A2HRH1TACR2
SCHEMBL10550052 0.86 POLB (0.47) KCNH2SSTR5NR4A2POLBHRH1
SCHEMBL9537249 0.86 SCN9A (0.53) KCNH2SSTR5NR4A2HRH1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed