SCHEMBL9537045

SCHEMBL9537045

O=Cc1ccc2cc3c(cc2c1)sc1ccccc13

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.44
KIF11 P52732 2/20 0.41
MAPT P10636 4/20 0.41
ALDH1A1 P00352 4/20 0.41
RAB9A P51151 4/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP2A6 P11509 6/20 0.40
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 1/20 0.39
PTPN7 P35236 1/20 0.37
DUSP3 P51452 1/20 0.37
PTPN12 Q05209 1/20 0.37
PTPN22 Q9Y2R2 1/20 0.37
CYP1A2 P05177 1/20 0.35
NPC1 O15118 2/20 0.35
KDM4E B2RXH2 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10970273 0.83 GPR3 (0.54) GPR3KIF11MAPTALDH1A1RAB9A
SCHEMBL6860177 0.83 GPR3 (0.54) GPR3KIF11MAPTALDH1A1RAB9A
SCHEMBL23513821 0.81 GPR3 (0.67) GPR3MAPTALDH1A1RAB9AHPGD
SCHEMBL23513817 0.81 GPR3 (0.67) GPR3MAPTALDH1A1RAB9AHPGD
SCHEMBL2336137 0.79 GPR3 (0.58) GPR3MAPTALDH1A1RAB9AHPGD
SCHEMBL23916960 0.79 GPR3 (0.64) GPR3MAPTALDH1A1RAB9AHPGD
SCHEMBL2742087 0.79 GPR3 (0.64) GPR3MAPTALDH1A1RAB9AHPGD
SCHEMBL29450187 0.79 GPR3 (0.64) GPR3MAPTALDH1A1RAB9AHPGD
SCHEMBL17356225 0.78 GPR3 (0.52) GPR3MAPTALDH1A1RAB9AHPGD
SCHEMBL17356251 0.78 GPR3 (0.52) GPR3MAPTALDH1A1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0182608-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-03-03 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4952597-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-08-28 US disclosed
US-4918101-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-04-17 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed
US-4873258-A Benzo[c] carbazole propanediol containing anti tumor compositions and use BURROUGHS WELLCOME CO. (US) 1989-10-10 US disclosed
US-4855453-A Tetracyclic thiophene derivatives BURROUGHS WELLCOME CO. (US) 1989-08-08 US disclosed
US-4797495-A ANTITUMOR AGENTS, ANTICARCINOGENIC AGENTS BURROUGHS WELLCOME CO. (US) 1989-01-10 US disclosed
EP-0182608-A2 Polycyclic compounds, their preparation and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-05-28 EP disclosed