SCHEMBL9537099

SCHEMBL9537099

CC(CO)(CO)NCc1cc2ccc3ccc4ccccc4c3c2o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.40
CYP2D6 P10635 2/20 0.35
MAPT P10636 4/20 0.34
ALDH1A1 P00352 4/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 2/20 0.34
THRB P10828 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
MPI P34949 1/20 0.34
KMT2A Q03164 3/20 0.32
NPBWR1 P48145 1/20 0.32
MCHR1 Q99705 1/20 0.32
PRKDC P78527 1/20 0.32
MEN1 O00255 2/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538254 0.94 SLC2A1 (0.48) SLC2A1CYP2D6MAPTALDH1A1L3MBTL1
SCHEMBL9526537 0.91 SLC2A1 (0.40) SLC2A1CYP2D6MAPTALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL9526852 0.90 SLC2A1 (0.39) SLC2A1CYP2D6MAPTALDH1A1L3MBTL1
SCHEMBL9535421 0.88 SLC2A1 (0.38) SLC2A1CYP2D6MAPTALDH1A1KDM4E
SCHEMBL9538259 0.86 SLC2A1 (0.40) SLC2A1CYP2D6MAPTALDH1A1L3MBTL1
SCHEMBL9779155 0.82 SLC2A1 (0.46) SLC2A1CYP2D6MAPTALDH1A1KDM4E
SCHEMBL9524760 0.80 KDM4E (0.46) SLC2A1MAPTALDH1A1L3MBTL1HSD17B10
SCHEMBL9535925 0.79 SLC2A1 (0.37) SLC2A1CYP1A2
Hydrochloric Acid SCHEMBL9526162 0.79 KDM4E (0.45) SLC2A1MAPTALDH1A1L3MBTL1HSD17B10
SCHEMBL9536493 0.78 ALDH1A1 (0.39) CYP2D6MAPTALDH1A1L3MBTL1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0182608-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-03-03 EP claimed
EP-0182608-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-03-03 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4952597-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-08-28 US disclosed
US-4918101-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-04-17 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed
US-4873258-A Benzo[c] carbazole propanediol containing anti tumor compositions and use BURROUGHS WELLCOME CO. (US) 1989-10-10 US disclosed
US-4855453-A Tetracyclic thiophene derivatives BURROUGHS WELLCOME CO. (US) 1989-08-08 US disclosed
US-4797495-A ANTITUMOR AGENTS, ANTICARCINOGENIC AGENTS BURROUGHS WELLCOME CO. (US) 1989-01-10 US disclosed
EP-0182608-A2 Polycyclic compounds, their preparation and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-05-28 EP disclosed