SCHEMBL9537117

SCHEMBL9537117

O=C(O)Cn1c(=O)c2cc(F)cnc2n(Cc2ccc(Br)cc2F)c1=O

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 9/20 0.60
AKR1A1 P14550 1/20 0.60
CYP1A2 P05177 2/20 0.48
CYP2C9 P11712 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48
AKR1B10 O60218 2/20 0.45
PTGDR2 Q9Y5Y4 2/20 0.43
TBXA2R P21731 1/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C8 P10632 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2A6 P11509 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTGDR Q13258 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535268 0.91 AKR1B1 (0.59) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL9535570 0.90 AKR1B1 (0.66) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL9534750 0.87 AKR1B1 (0.55) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL9535225 0.85 AKR1B1 (0.60) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL10487878 0.79 AKR1B1 (0.86) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL9319101 0.79 AKR1B1 (0.81) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL10487918 0.78 AKR1B1 (0.76) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL9056716 0.77 AKR1B1 (0.78) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL10487834 0.76 AKR1B1 (0.79) AKR1B1AKR1A1CYP1A2CYP2C9MEN1
SCHEMBL10487869 0.75 AKR1B1 (0.78) AKR1B1AKR1A1CYP1A2CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0568540-A1 2,4-DIOXO-PYRIDO 2,3-d]PYRIMIDINE-3-ACETIC ACIDS AND ESTERS AND SALTS THEREOF PFIZER INC. (US) 1993-11-10 EP disclosed
WO-1992012979-A1 2,4-DIOXO-PYRIDO [2,3-d]PYRIMIDINE-3-ACETIC ACIDS AND ESTERS AND SALTS THEREOF PFIZER INC. (US) 1992-08-06 WO disclosed