SCHEMBL9537137

SCHEMBL9537137

Oc1ccc2c(c1)CC(NCC(O)COc1cccc(Cl)c1)CC2

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 11/20 0.56
ADRB1 P08588 3/20 0.56
NPY1R P25929 1/20 0.53
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
THPO P40225 1/20 0.49
NPC1 O15118 1/20 0.49
MTOR P42345 1/20 0.49
RAB9A P51151 1/20 0.49
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9587385 0.99 ADRB3 (0.55) ADRB3ADRB1NPY1RTP53CYP1A2
SCHEMBL9535995 0.91 NPY1R (0.65) ADRB3ADRB1NPY1RTP53CYP1A2
Hydrochloric Acid SCHEMBL9586636 0.90 NPY1R (0.64) ADRB3ADRB1NPY1RTP53CYP1A2
SCHEMBL9533941 0.89 NPY1R (0.65) ADRB3ADRB1NPY1RTP53CYP1A2
Hydrochloric Acid SCHEMBL9587899 0.88 NPY1R (0.64) ADRB3ADRB1NPY1RTP53CYP1A2
SCHEMBL9535842 0.86 TP53 (0.46) ADRB3ADRB1NPY1RTP53CYP1A2
SCHEMBL9536728 0.86 NPY1R (0.53) ADRB3ADRB1NPY1RTP53CYP1A2
Hydrochloric Acid SCHEMBL9587656 0.85 TP53 (0.46) ADRB3ADRB1NPY1RTP53CYP1A2
Hydrochloric Acid SCHEMBL9587381 0.85 NPY1R (0.52) ADRB3ADRB1NPY1RTP53CYP1A2
SCHEMBL22279183 0.83 ADRB3 (0.51) ADRB3ADRB1NPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed