SCHEMBL9537507

SCHEMBL9537507

CC(CO)(CO)NCc1c2ccccc2cc2oc3ccccc3c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.38
ADRB2 P07550 1/20 0.37
NPBWR1 P48145 1/20 0.34
KMT2A Q03164 1/20 0.34
MCHR1 Q99705 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CD274 Q9NZQ7 1/20 0.33
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAOA P21397 2/20 0.33
GAA P10253 2/20 0.32
MGAM O43451 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
ALDH1A1 P00352 2/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535779 0.94 SLC2A1 (0.46) SLC2A1ADRB2NPBWR1KMT2AMCHR1
SCHEMBL9535783 0.86 SLC2A1 (0.38) SLC2A1ADRB2NPBWR1KMT2AMCHR1
SCHEMBL9843654 0.85 SLC2A1 (0.35) SLC2A1ADRB2L3MBTL1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL9843354 0.84 SLC2A1 (0.35) SLC2A1ADRB2KMT2AL3MBTL1CD274
SCHEMBL9536399 0.82 SLC2A1 (0.36) SLC2A1NPBWR1KMT2AMCHR1RAB9A
SCHEMBL10488406 0.81 HTR2A (0.43) SLC2A1NPBWR1KMT2AMCHR1L3MBTL1
Hydrochloric Acid SCHEMBL10488372 0.80 KMT2A (0.43) SLC2A1NPBWR1KMT2AMCHR1L3MBTL1
SCHEMBL9536568 0.80 SLC2A1 (0.49) SLC2A1ADRB2KMT2AL3MBTL1RAB9A
SCHEMBL9537834 0.78 SLC2A1 (0.44) SLC2A1NPBWR1KMT2AMCHR1RAB9A
SCHEMBL9526392 0.78 ADRB2 (0.43) SLC2A1ADRB2RAB9ASMN1; SMN2CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0182608-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-03-03 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4952597-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-08-28 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed
US-4873258-A Benzo[c] carbazole propanediol containing anti tumor compositions and use BURROUGHS WELLCOME CO. (US) 1989-10-10 US disclosed
US-4855453-A Tetracyclic thiophene derivatives BURROUGHS WELLCOME CO. (US) 1989-08-08 US disclosed
US-4797495-A ANTITUMOR AGENTS, ANTICARCINOGENIC AGENTS BURROUGHS WELLCOME CO. (US) 1989-01-10 US disclosed
EP-0182608-A2 Polycyclic compounds, their preparation and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-05-28 EP disclosed