SCHEMBL9537797

SCHEMBL9537797

[CH2]CN1CCC(Cc2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.57
SSTR5 P35346 3/20 0.53
CYP2D6 P10635 7/20 0.52
HRH1 P35367 7/20 0.52
KCNH2 Q12809 5/20 0.52
CHRM1 P11229 3/20 0.52
HTR3A P46098 1/20 0.48
NR1I2 O75469 1/20 0.48
ABCB11 O95342 1/20 0.48
LMNA P02545 1/20 0.48
ESR1 P03372 1/20 0.48
CYP1A2 P05177 1/20 0.48
PGR P06401 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
TSHR P16473 1/20 0.48
ADRA2B P18089 1/20 0.48
HTR2A P28223 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536543 0.90 SSTR5 (0.66) RAB9ASSTR5CYP2D6HRH1KCNH2
SCHEMBL9536663 0.87 RAB9A (0.55) RAB9ASSTR5CYP2D6HRH1KCNH2
Hydrochloric Acid SCHEMBL9537670 0.87 RAB9A (0.55) RAB9ASSTR5CYP2D6HRH1KCNH2
SCHEMBL9537554 0.87 HRH1 (0.63) RAB9ASSTR5CYP2D6HRH1KCNH2
SCHEMBL9536935 0.86 NPSR1 (0.55) RAB9ASSTR5CYP2D6HRH1KCNH2
Hydrochloric Acid SCHEMBL9539517 0.86 HRH1 (0.62) RAB9ASSTR5CYP2D6HRH1KCNH2
Hydrochloric Acid SCHEMBL9537718 0.85 TP53 (0.52) RAB9ASSTR5CYP2D6HRH1KCNH2
SCHEMBL9539669 0.85 RAB9A (0.52) RAB9ASSTR5CYP2D6HRH1KCNH2
SCHEMBL9537249 0.85 SCN9A (0.53) RAB9ASSTR5CYP2D6HRH1KCNH2
SCHEMBL9537151 0.85 SSTR5 (0.59) RAB9ASSTR5CYP2D6HRH1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed