SCHEMBL9537829

SCHEMBL9537829

COc1ccc2nc(CC3CCNCC3)n(Cc3ccc(F)cc3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.58
NR4A2 P43354 1/20 0.45
SSTR5 P35346 1/20 0.44
SOS1 Q07889 1/20 0.43
HTR3A P46098 1/20 0.43
RAB9A P51151 1/20 0.42
TBXA2R P21731 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9539127 0.90 KCNH2 (0.56) KCNH2NR4A2SSTR5SOS1HTR3A
SCHEMBL9538624 0.88 KCNH2 (0.63) KCNH2NR4A2SOS1HTR3ARAB9A
SCHEMBL9537805 0.85 SSTR5 (0.56) KCNH2SSTR5HTR3ATBXA2R
SCHEMBL9535886 0.85 KCNH2 (0.59) KCNH2NR4A2SOS1HTR3ARAB9A
SCHEMBL10548476 0.84 KCNH2 (0.62) KCNH2NR4A2SOS1RAB9A
SCHEMBL10551636 0.84 KCNH2 (0.62) KCNH2NR4A2SOS1RAB9A
SCHEMBL9537539 0.83 HTR3A (0.62) KCNH2HTR3ATBXA2R
Oxalic Acid SCHEMBL10549909 0.82 KCNH2 (0.56) KCNH2NR4A2SOS1TBXA2R
Oxalic Acid SCHEMBL10549899 0.82 KCNH2 (0.56) KCNH2NR4A2SOS1TBXA2R
SCHEMBL9382803 0.82 KCNH2 (0.64) KCNH2NR4A2HTR3ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed