SCHEMBL9538555

SCHEMBL9538555

Cc1c[nH]c(=S)c(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMBS P08397 1/20 0.41
ALDH1A1 P00352 8/20 0.37
MAPT P10636 5/20 0.37
RXFP1 Q9HBX9 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HAVCR2 Q8TDQ0 1/20 0.37
HPGD P15428 5/20 0.37
APOBEC3G Q9HC16 3/20 0.37
KDM4E B2RXH2 3/20 0.36
ALOX12 P18054 2/20 0.36
ALOX15 P16050 2/20 0.36
HSD17B10 Q99714 2/20 0.36
MCL1 Q07820 1/20 0.36
POLB P06746 1/20 0.34
DAO P14920 1/20 0.32
DPYD Q12882 1/20 0.31
LRRK2 Q5S007 2/20 0.31
TSHR P16473 1/20 0.31
HSP90AB1 P08238 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3828174 0.77 ALDH1A1 (0.38) ALDH1A1MAPTRXFP1MEN1KMT2A
SCHEMBL9356587 0.75 MCL1 (0.58) HMBSALDH1A1HPGDKDM4EMCL1
SCHEMBL8646977 0.71 ALDH1A1 (0.37) ALDH1A1MAPTRXFP1MEN1KMT2A
SCHEMBL10963619 0.66 CYP19A1 (0.41) ALDH1A1MAPTMEN1KMT2AHPGD
SCHEMBL21596508 0.66
SCHEMBL11948728 0.64 TSHR (0.40) ALDH1A1MAPTKMT2AKDM4EALOX15
SCHEMBL11445453 0.62 TSHR (0.39) ALDH1A1MAPTMEN1KMT2AHAVCR2
SCHEMBL3214424 0.61 DPYD (0.34) ALDH1A1MAPTRXFP1MEN1KMT2A
SCHEMBL2977054 0.61
SCHEMBL1003862 0.61 ALDH1A1 (0.46) ALDH1A1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215063-B1 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES UNIV PRINCETON (US) 1993-11-03 EP disclosed
US-5026851-A Antineoplastic agents THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-25 US disclosed
US-4845216-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-07-04 US disclosed
EP-0215063-A4 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES. UNIV PRINCETON (US) 1987-11-23 EP disclosed
US-4684653-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1987-08-04 US disclosed
EP-0215063-A1 PYRIDO (2,3-d )PYRIMIDIN DERIVATIVES. UNIV PRINCETON (US) 1987-03-25 EP disclosed
WO-1986005181-A1 PYRIDO AD2,3-d BDPYRIMIDIN DERIVATIVES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1986-09-12 WO disclosed