SCHEMBL9538592

SCHEMBL9538592

[c]1c(-c2cccnc2)ccnc1-c1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 11/20 0.50
ALDH1A1 P00352 3/20 0.50
CYP3A4 P08684 3/20 0.50
CYP1A2 P05177 2/20 0.50
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PTK2 Q05397 1/20 0.42
MEN1 O00255 1/20 0.42
PSIP1 O75475 1/20 0.42
AXL P30530 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434201 0.76 ASIC3 (0.44) ALDH1A1SMN1; SMN2HSP90AA1PTK2DYRK1B
SCHEMBL2112813 0.72 CYP2A6 (0.52) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL973260 0.72 CYP2A6 (0.53) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL120088 0.70 CYP2A6 (1.00) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL29419014 0.70 CYP2A6 (1.00) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL30473120 0.70 CYP2A6 (1.00) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL21295738 0.69 CYP2A6 (0.44) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL12108682 0.68 CYP2A6 (0.83) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL12956908 0.68 CYP2A6 (0.83) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL31508264 0.68 CYP2A6 (0.83) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543930-A1 ARTHROPODICIDAL PYRAZOLINES, PYRAZOLIDINES AND HYDRAZINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-06-02 EP disclosed
WO-1992003421-A2 ARTHROPODICIDAL PYRAZOLINES, PYRAZOLIDINES AND HYDRAZINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-03-05 WO disclosed