SCHEMBL9538640

SCHEMBL9538640

CC(CO)(CO)NCc1cc2c3ccccc3ccc2c2sccc12

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.58
CSNK2A1 P68400 10/20 0.33
CYP1A2 P05177 1/20 0.32
NPBWR1 P48145 1/20 0.31
KMT2A Q03164 1/20 0.31
MCHR1 Q99705 1/20 0.31
MAPK8 P45983 2/20 0.31
MAPK9 P45984 1/20 0.31
MAPK10 P53779 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
HPRT1 P00492 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538875 0.95 SLC2A1 (0.67) SLC2A1CSNK2A1MAPK8MAPK9MAPK10
SCHEMBL9538878 0.87 SLC2A1 (0.55) SLC2A1
Crisnatol SCHEMBL15990 0.85 SLC2A1 (0.52) SLC2A1CYP1A2NPBWR1KMT2AMCHR1
Crisnatol SCHEMBL6257042 0.85 SLC2A1 (0.52) SLC2A1CYP1A2NPBWR1KMT2AMCHR1
Crisnatol SCHEMBL10484286 0.84 SLC2A1 (0.51) SLC2A1CYP1A2NPBWR1KMT2AMCHR1
SCHEMBL9779055 0.83 SLC2A1 (0.69) SLC2A1CYP1A2
SCHEMBL9524655 0.82 SLC2A1 (0.70) SLC2A1CYP1A2ALDH1A1HPGD
SCHEMBL9779019 0.81 SLC2A1 (0.53) SLC2A1CYP1A2NPBWR1KMT2AMCHR1
Hydrochloric Acid SCHEMBL9764686 0.81 SLC2A1 (0.48) SLC2A1CYP1A2NPBWR1KMT2AMCHR1
Hydrochloric Acid SCHEMBL9525862 0.81 SLC2A1 (0.69) SLC2A1CYP1A2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0182608-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-03-03 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4952597-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-08-28 US disclosed
US-4918101-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-04-17 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed
US-4873258-A Benzo[c] carbazole propanediol containing anti tumor compositions and use BURROUGHS WELLCOME CO. (US) 1989-10-10 US disclosed
US-4855453-A Tetracyclic thiophene derivatives BURROUGHS WELLCOME CO. (US) 1989-08-08 US disclosed
US-4797495-A ANTITUMOR AGENTS, ANTICARCINOGENIC AGENTS BURROUGHS WELLCOME CO. (US) 1989-01-10 US disclosed
EP-0182608-A2 Polycyclic compounds, their preparation and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-05-28 EP disclosed