SCHEMBL9540106

SCHEMBL9540106

CCC1(c2ccccc2)c2cc(Cl)ccc2NC(=S)N1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PGR P06401 8/20 0.40
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
ALOX12 P18054 1/20 0.38
KMT2A Q03164 1/20 0.38
CHRM1 P11229 10/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539014 0.86 AKR1B1 (0.40) PGRMEN1MAPTKMT2ACHRM1
SCHEMBL9539805 0.85 PGR (0.41) PGRKDM4EMEN1ALDH1A1MAPT
SCHEMBL9542468 0.84 PGR (0.40) PGRKDM4EMEN1ALDH1A1MAPT
SCHEMBL9539046 0.78 PGR (0.38) PGRMAPTCHRM1
SCHEMBL9539937 0.78 CHRM1 (0.41) PGRKDM4EMEN1ALDH1A1MAPT
SCHEMBL9539997 0.77 PGR (0.39) PGRALDH1A1MAPTALOX12CHRM1
SCHEMBL9540047 0.76 PGR (0.40) PGRKDM4EMEN1ALDH1A1MAPT
SCHEMBL9539803 0.76 PGR (0.38) PGRKDM4EALDH1A1MAPTCHRM1
SCHEMBL9539722 0.75 AKR1B1 (0.50) PGRMAPT
SCHEMBL4594261 0.74 AKR1B1 (0.43) PGRMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed