SCHEMBL9540132

SCHEMBL9540132

COc1ccc(CN2C(=O)NC(C)(C(C)C)c3ccccc32)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.54
CASP3 P42574 1/20 0.47
OPRL1 P41146 1/20 0.47
CMA1 P23946 1/20 0.47
MMP12 P39900 1/20 0.46
ADAMTS5 Q9UNA0 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
MAPT P10636 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
HTT P42858 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
EDNRB P24530 1/20 0.42
EDNRA P25101 1/20 0.42
PIM1 P11309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14501653 0.85 SCN9A (0.55) SCN9ACASP3OPRL1CMA1MMP12
SCHEMBL16109588 0.81 SCN9A (0.56) SCN9ACMA1MMP12ADAMTS5L3MBTL1
SCHEMBL9539012 0.80 OPRL1 (0.51) SCN9ACASP3OPRL1CMA1MMP12
SCHEMBL17377477 0.77 SCN9A (0.63) SCN9ACASP3OPRL1CMA1MMP12
SCHEMBL25430199 0.76 SCN9A (0.65) SCN9ACASP3OPRL1CMA1MMP12
SCHEMBL17416402 0.73 OPRL1 (0.70) SCN9AOPRL1CMA1MMP12ADAMTS5
SCHEMBL15973283 0.72 SCN9A (0.51) SCN9ACASP3CMA1MMP12ADAMTS5
SCHEMBL16812434 0.72 OPRL1 (0.60) SCN9ACASP3OPRL1CMA1MMP12
SCHEMBL8552517 0.72 SCN9A (0.54) SCN9ACASP3OPRL1CMA1MMP12
SCHEMBL1773322 0.71 CMA1 (0.60) CASP3CMA1L3MBTL1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed