SCHEMBL9541141

SCHEMBL9541141

CC(=O)O[C@@]1(C)CC[C@H]2[C@@H]3CC=C4C=C(N5CCCC5)CC[C@]4(C)[C@H]3CC[C@@]21C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.47
SRD5A2 P31213 9/20 0.41
ESR1 P03372 2/20 0.39
AR P10275 2/20 0.39
ESR2 Q92731 2/20 0.39
LMNA P02545 2/20 0.38
CYP3A4 P08684 2/20 0.38
ABCC4 O15439 1/20 0.38
ABCB11 O95342 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NR3C1 P04150 1/20 0.38
SHBG P04278 1/20 0.38
PGR P06401 1/20 0.38
CHRM2 P08172 1/20 0.38
NR3C2 P08235 1/20 0.38
CHRM1 P11229 1/20 0.38
HRH2 P25021 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24358654 0.84 SHBG (0.53) CYP17A1SRD5A2ESR1ARESR2
SCHEMBL9195965 0.84 SHBG (0.53) CYP17A1SRD5A2ESR1ARESR2
SCHEMBL24358655 0.84 SHBG (0.53) CYP17A1SRD5A2ESR1ARESR2
SCHEMBL9543900 0.83 SHBG (0.49) SRD5A2ESR1ARESR2LMNA
SCHEMBL24358694 0.78 SRD5A2 (0.59) SRD5A2ESR1ARESR2LMNA
SCHEMBL11731128 0.78 SHBG (0.53) ESR1ARESR2LMNACYP3A4
SCHEMBL11326365 0.78 CYP19A1 (0.57) SRD5A2LMNACYP3A4SHBGCYP19A1
SCHEMBL11643796 0.76 ESR1 (0.41) SRD5A2ESR1ARESR2LMNA
SCHEMBL11207949 0.73 SRD5A2 (0.43) SRD5A2ESR1ARESR2LMNA
SCHEMBL11343684 0.71 TDP1 (0.40) SRD5A2ESR1ARESR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013122-A1 3-METHYLSULPHONYLHYDRAZONO AND 3-OXYIMINO STEROIDS, A METHOD OF PREPARING THEM, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND THEIR USE IN THE PREPARATION OF DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1993-07-08 WO disclosed