SCHEMBL9541557

SCHEMBL9541557

CCOCCC1(C2CC2)c2cc(Cl)ccc2NC(=O)N1CC

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AKR1B1 P15121 3/20 0.36
MMP14 P50281 4/20 0.35
HTR7 P34969 3/20 0.35
IDO1 P14902 1/20 0.34
ELOVL6 Q9H5J4 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
MMP13 P45452 2/20 0.34
CYP46A1 Q9Y6A2 1/20 0.34
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
PDE7A Q13946 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539091 0.91 MEN1 (0.39) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL9540069 0.87 MEN1 (0.41) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL9539784 0.85 MEN1 (0.40) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL9539061 0.77 MEN1 (0.39) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL9539065 0.76 AKR1B1 (0.45) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL2473132 0.76 AKR1B1 (0.40) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL2471933 0.75 HTR7 (0.38) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL9539079 0.74 AKR1B1 (0.48) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL2467635 0.74 CYP46A1 (0.39) MEN1KMT2AAKR1B1HTR7IDO1
SCHEMBL2471338 0.74 CYP46A1 (0.37) MEN1KMT2AAKR1B1HTR7IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed