SCHEMBL9542390

SCHEMBL9542390

N#CC1(N)CCN(Cc2ccccc2)CC1.NC1(C(=O)O)CCN(Cc2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.53
TSHR P16473 3/20 0.48
CYP2D6 P10635 6/20 0.48
CHRM2 P08172 3/20 0.47
CHRM3 P20309 1/20 0.47
OPRL1 P41146 2/20 0.47
ALDH1A1 P00352 3/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 5/20 0.46
HSD17B10 Q99714 1/20 0.46
USP2 O75604 2/20 0.44
MAPK1 P28482 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
CYP2C19 P33261 1/20 0.43
GRM6 O15303 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CCR3 P51677 1/20 0.43
CHRM4 P08173 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1587072 0.89 OPRM1 (0.65) OPRM1TSHRCYP2D6OPRL1ALDH1A1
SCHEMBL1975609 0.89 CYP2D6 (0.57) TSHRCYP2D6CHRM2CHRM3OPRL1
Hydrochloric Acid SCHEMBL10732688 0.87 POLB (0.58) TSHRCYP2D6CHRM2CHRM3OPRL1
Hydrochloric Acid SCHEMBL2088271 0.87 POLB (0.58) TSHRCYP2D6CHRM2CHRM3OPRL1
Sulfuric Acid SCHEMBL11839097 0.83 MAPK1 (0.56) TSHRCYP2D6CHRM2CHRM3OPRL1
SCHEMBL9542332 0.83 OPRM1 (0.55) OPRM1TSHRCYP2D6OPRL1ALDH1A1
SCHEMBL3893581 0.80 OPRM1 (0.57) OPRM1TSHRCYP2D6OPRL1ALDH1A1
SCHEMBL8576692 0.80 CYP2D6 (0.55) TSHRCYP2D6CHRM2CHRM3OPRL1
Bromide SCHEMBL8574506 0.79 CYP2D6 (0.54) TSHRCYP2D6CHRM2CHRM3OPRL1
SCHEMBL3955531 0.79 TSHR (0.63) TSHRCYP2D6CHRM2CHRM3OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993000359-A1 MODIFIED PEPTIDES TRANSPORTABLE INTO THE CENTRAL NERVOUS SYSTEM THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-01-07 WO disclosed