SCHEMBL9542596

SCHEMBL9542596

N#Cc1ccccc1-c1ccc(CI)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.59
FFAR1 O14842 1/20 0.47
AKR1B1 P15121 1/20 0.47
PTPN5 P54829 1/20 0.46
PPARG P37231 2/20 0.45
GSK3B P49841 2/20 0.45
GSK3A P49840 1/20 0.45
PRKAG1 P54619 3/20 0.44
PRKAA1 Q13131 3/20 0.44
PRKAB1 Q9Y478 3/20 0.44
ACHE P22303 1/20 0.44
MME P08473 1/20 0.44
CNR2 P34972 1/20 0.44
TRPA1 O75762 1/20 0.42
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
PDE10A Q9Y233 1/20 0.40
MYC P01106 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1713 0.83 ESR2 (0.67) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL31410710 0.82 ESR2 (0.76) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL29170999 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL357 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL360601 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL31772593 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL3169219 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL7867991 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL31124937 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG
SCHEMBL26016200 0.81 ESR2 (0.59) ESR2FFAR1AKR1B1PTPN5PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed