SCHEMBL9543386

SCHEMBL9543386

Oc1ccc(CCNCC(O)c2ccccc2)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.73
KDM4E B2RXH2 2/20 0.63
GAA P10253 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
TDP1 Q9NUW8 1/20 0.63
ADRB3 P13945 8/20 0.60
L3MBTL1 Q9Y468 1/20 0.59
ADRB1 P08588 3/20 0.59
ALDH1A1 P00352 1/20 0.59
LMNA P02545 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
SLC22A1 O15245 1/20 0.59
CHRM2 P08172 1/20 0.59
CYP3A4 P08684 1/20 0.59
CHRM1 P11229 1/20 0.59
TSHR P16473 1/20 0.59
NFKB1 P19838 1/20 0.59
SLC6A4 P31645 1/20 0.59
OPRM1 P35372 1/20 0.59
SLC6A3 Q01959 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4467889 1.00 ADRB2 (0.73) ADRB2KDM4EGAASMN1; SMN2TDP1
SCHEMBL4467885 1.00 ADRB2 (0.73) ADRB2KDM4EGAASMN1; SMN2TDP1
SCHEMBL9467104 0.95 ADRB2 (0.68) ADRB2KDM4EGAASMN1; SMN2TDP1
SCHEMBL11467407 0.91 ADRB2 (0.61) ADRB2KDM4EGAASMN1; SMN2TDP1
SCHEMBL11467406 0.91 ADRB2 (0.61) ADRB2KDM4EGAASMN1; SMN2TDP1
SCHEMBL10720145 0.90 ADRB2 (0.77) ADRB2KDM4EGAASMN1; SMN2TDP1
Bromide SCHEMBL11470044 0.89 ADRB2 (0.59) ADRB2KDM4EGAASMN1; SMN2TDP1
Bromide SCHEMBL11470045 0.89 ADRB2 (0.59) ADRB2KDM4EGAASMN1; SMN2TDP1
SCHEMBL19245594 0.86 ADRB2 (0.71) ADRB2KDM4EGAASMN1; SMN2TDP1
SCHEMBL19245591 0.86 ADRB2 (0.71) ADRB2KDM4EGAASMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101516826-A Beta-3 receptor ligands and therapeutic uses thereof UNIV BARI (IT) 2009-08-26 CN claimed
CN-101516826-B Beta-3 receptor ligands UNIV BARI 2015-03-04 CN disclosed
CN-101516826-A Beta-3 receptor ligands and therapeutic uses thereof UNIV BARI (IT) 2009-08-26 CN disclosed
WO-1993010074-A1 ARYLETHANOLAMINE DERIVATIVES AND THEIR USE AS BETA-3-ADRENOCEPTOR AGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-05-27 WO disclosed