SCHEMBL9543765

SCHEMBL9543765

CC1=C2CC[C@@H]3[C@H](CC[C@@]4(C)[C@H]3CC[C@@]4(O)C#CCl)[C@@]2(C)CC/C1=N\O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHBG P04278 4/20 0.41
TSHR P16473 4/20 0.41
HIF1A Q16665 4/20 0.41
ESR1 P03372 3/20 0.41
NR3C1 P04150 3/20 0.41
PGR P06401 3/20 0.41
CYP2C19 P33261 3/20 0.41
LMNA P02545 3/20 0.41
THRB P10828 1/20 0.41
MEN1 O00255 1/20 0.41
AR P10275 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP3A4 P08684 5/20 0.40
PDK1 Q15118 1/20 0.37
PDK2 Q15119 1/20 0.37
PDK3 Q15120 1/20 0.37
PDK4 Q16654 1/20 0.37
THPO P40225 2/20 0.35
TDP1 Q9NUW8 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542060 0.87 SHBG (0.54) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9541208 0.85 CYP3A4 (0.58) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9541949 0.85 SHBG (0.38) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9541880 0.85 SHBG (0.38) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9541942 0.83 SHBG (0.50) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9542589 0.75 SHBG (0.39) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL11520495 0.75 CYP3A4 (0.59) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9542845 0.75 SHBG (0.60) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9541266 0.74 CYP17A1 (0.51) SHBGTSHRHIF1AESR1NR3C1
SCHEMBL9542422 0.74 CYP3A4 (0.39) SHBGTSHRHIF1AESR1NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013122-A1 3-METHYLSULPHONYLHYDRAZONO AND 3-OXYIMINO STEROIDS, A METHOD OF PREPARING THEM, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND THEIR USE IN THE PREPARATION OF DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1993-07-08 WO claimed
WO-1993013122-A1 3-METHYLSULPHONYLHYDRAZONO AND 3-OXYIMINO STEROIDS, A METHOD OF PREPARING THEM, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND THEIR USE IN THE PREPARATION OF DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1993-07-08 WO disclosed