SCHEMBL9544430

SCHEMBL9544430

Cc1ccc(C2CC2C#N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
FFAR1 O14842 1/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CYP2A6 P11509 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
PRNP P04156 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
BRCA1 P38398 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31611782 0.82 HTR2A (0.39) HTR2AHTR2CHTR2BFFAR1ALDH1A1
SCHEMBL18704254 0.79 HTR2A (0.44) HTR2AHTR2CHTR2BCYP2A6MAPT
SCHEMBL5310780 0.79 KDM1A (0.52) HTR2CHTR2BCYP2C9CYP2C19CYP2A6
SCHEMBL2359930 0.79 FFAR1 (0.45) HTR2AHTR2CHTR2BFFAR1ALDH1A1
SCHEMBL9543138 0.79 KDM1A (0.56) HTR2CKDM4EMEN1MAPTKMT2A
SCHEMBL8136211 0.79 GRIA4 (0.39) HTR2AHTR2CHTR2BFFAR1ALDH1A1
SCHEMBL8579770 0.79 GRIA4 (0.39) HTR2AHTR2CHTR2BFFAR1ALDH1A1
SCHEMBL8830861 0.79 HTR2A (0.37) HTR2AHTR2CHTR2BFFAR1ALDH1A1
SCHEMBL5450245 0.78 MAOB (0.48) HTR2AHTR2CHTR2BCYP1A2CYP3A4
SCHEMBL3946310 0.72 TAAR1 (0.38) HTR2AALDH1A1CYP1A2CYP2C19CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993015100-A1 NOVEL ADENOSINE DERIVATIVES, THEIR PREPARATION METHODS AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LABORATOIRES UPSA (FR) 1993-08-05 WO disclosed